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>【930】去甲肾上腺素临床应用要点.ppt
【930】去甲肾上腺素临床应用要点.ppt
2026-05-11 01:05:45
【930】去甲肾上腺素临床应用要点.ppt
需要公众号里的ppt,点我咨询~
先看看我写的学习笔记,PPT往下翻。
一、基本药理
1. 基本信息
类别:儿茶酚胺类神经递质、激素,肾上腺素合成前体
临床制剂:重酒石酸去甲肾上腺素
分泌来源:交感神经末梢、肾上腺髓质
2. 结构与药理作用
结构:含邻苯二酚环与乙胺侧链
作用:强效激动 α 受体,弱激动 β₁受体,几乎不激动 β₂受体
3. 受体效应
α 受体:收缩小动脉、静脉,升高外周阻力
β₁受体:轻度增强心肌收缩力、加快心率、加速传导
β₂受体:无明显激动效应,不引起血管扩张
二、适应症与用法用量
1. 适应症
急性心肌梗死、体外循环所致低血压
血容量不足性休克、嗜铬细胞瘤术后低血压
椎管内阻滞低血压、心脏停搏复苏后血压维持
感染性休克升压支持
口服用于上消化道出血
2. 用法用量
低血压、休克
静脉滴注:起始 8~12μg/min,维持 2~4μg/min,上限不超过 25μg/min
危急静注:1~2mg 稀释至 10~20mL 缓慢推注,后继以滴注维持
上消化道出血
口服:1~3mg / 次,加冷盐水送服,每日 3 次
三、溶媒选择
1. 稳定性特点
易氧化,碱性环境加速降解,微酸性稳定
2. 推荐溶媒
首选:5% 葡萄糖注射液、葡萄糖氯化钠注射液
替代:生理盐水可现配现用
四、与肾上腺素的区别
1. 结构差异
去甲肾上腺素:侧链氨基为 - NH₂
肾上腺素:侧链氨基为 - NHCH₃
2. 受体作用
去甲肾上腺素:α 强、β₁弱、β₂无
肾上腺素:α 极强、β₁强、β₂强
3. 临床用途
去甲肾上腺素:休克升压、低血压维持
肾上腺素:过敏性休克、心肺复苏
五、药物相互作用
全麻药、洋地黄、三环类抗抑郁药:易致心律失常,需小剂量、监护
β 受体阻滞药:α 作用占优,可致高血压、心动过缓
降压药:作用抵消,避免联用
麦角制剂、缩宫素:血管过度收缩,禁用
甲状腺激素:作用均增强,慎用
六、应用注意事项
1. 特殊人群
妊娠期:减少子宫血流,胎儿缺氧风险,慎用
2. 局部风险
药液外漏、浓度过高可致组织坏死
处理:酚妥拉明 5~10mg 稀释后局部浸润注射
3. 肾功能风险
大剂量、长期使用可致肾血管收缩、无尿、肾损伤
监测尿量与肾功能
七、小结
以 α 收缩血管为主,β₁轻度强心,用于重症升压
优先葡萄糖溶媒,严防外渗,监测尿量与心率
联用需谨慎,禁忌与麦角类、强效降压药合用
兼顾升压效果与心、肾、肢体灌注安全
需要公众号里的ppt,点我咨询~
需要公众号里的ppt,点我咨询~
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CONNECT:[ UseTime:0.001019s ] mysql:host=127.0.0.1;port=3306;dbname=h_sjds;charset=utf8mb4
SHOW FULL COLUMNS FROM `fenlei` [ RunTime:0.001924s ]
SELECT * FROM `fenlei` WHERE `fid` = 0 [ RunTime:0.000794s ]
SELECT * FROM `fenlei` WHERE `fid` = 63 [ RunTime:0.000646s ]
SHOW FULL COLUMNS FROM `set` [ RunTime:0.001536s ]
SELECT * FROM `set` [ RunTime:0.000598s ]
SHOW FULL COLUMNS FROM `article` [ RunTime:0.001550s ]
SELECT * FROM `article` WHERE `id` = 512503 LIMIT 1 [ RunTime:0.002228s ]
UPDATE `article` SET `lasttime` = 1778759428 WHERE `id` = 512503 [ RunTime:0.029410s ]
SELECT * FROM `fenlei` WHERE `id` = 64 LIMIT 1 [ RunTime:0.000837s ]
SELECT * FROM `article` WHERE `id` < 512503 ORDER BY `id` DESC LIMIT 1 [ RunTime:0.001328s ]
SELECT * FROM `article` WHERE `id` > 512503 ORDER BY `id` ASC LIMIT 1 [ RunTime:0.007662s ]
SELECT * FROM `article` WHERE `id` < 512503 ORDER BY `id` DESC LIMIT 10 [ RunTime:0.002844s ]
SELECT * FROM `article` WHERE `id` < 512503 ORDER BY `id` DESC LIMIT 10,10 [ RunTime:0.000855s ]
SELECT * FROM `article` WHERE `id` < 512503 ORDER BY `id` DESC LIMIT 20,10 [ RunTime:0.003836s ]
0.244546s